抑制剂与激动剂

Catalog_noADMC0461
Product_nameAnamorelin
Category抑制剂与激动剂
Size10mg/50mg/100mg
Price1120.00/2120.00/2780.00
SpecificityTarget: GHSR. Fields: Anamorelin(RC1291; ONO-7643) is a synthetic orally active ghrelin receptor agonist which is under development for the management of non-small lung cancer associated cachexia/anorexia. Ki: 0.7 nM (ghrelin receptor)[1]EC50: 0.74
DilutionKi: 0.7 nM (ghrelin receptor)[1]EC50: 0.74 nM (ghrelin receptor)[1]
Purification>98%
Concentration靶点:GHSR;IC50:Ki: 0.7 nM (ghrelin receptor)[1]EC50: 0.74 nM (ghrelin receptor)[1]
Storage_stability2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
othernameRC-1291; ONO-7643; RC1291; ONO7643; RC 1291; ONO 7643
Observed_band546.7
NotesAnamorelin(RC1291; ONO-7643) is a synthetic orally active ghrelin receptor agonist which is under development for the management of non-small lung cancer associated cachexia/anorexia. Ki: 0.7 nM (ghrelin receptor)[1]EC50: 0.74 nM (ghrelin receptor)[1
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